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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM372279'
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt University

US Patent
LigandPNGBDBM372279(4-(azetidin-1-yl)-8- methylpyrido[3',2':4,5] thien...)
Affinity DataEC50:  2.50E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM372279(4-(azetidin-1-yl)-8- methylpyrido[3',2':4,5] thien...)
Affinity DataEC50:  807nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent