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Found 6 Enz. Inhib. hit(s) with Target = 'N-formyl peptide receptor 2' and Ligand = 'BDBM50520820'
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520820(CHEMBL4551559)
Affinity DataIC50:  3.40nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520820(CHEMBL4551559)
Affinity DataIC50:  3.70nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520820(CHEMBL4551559)
Affinity DataIC50:  4.30nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520820(CHEMBL4551559)
Affinity DataIC50:  4.80nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520820(CHEMBL4551559)
Affinity DataIC50:  40nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation pretreated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520820(CHEMBL4551559)
Affinity DataIC50:  56nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed