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Found 3 Enz. Inhib. hit(s) with Target = 'Neuromedin-K receptor' and Ligand = 'BDBM362839'
TargetNeuromedin-K receptor(Homo sapiens (Human))
Oged

US Patent
LigandPNGBDBM362839((R)-(4-fluorophenyl)(8- methyl-3-(5-methylfuran-2-...)
Affinity DataKi:  48nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeuromedin-K receptor(Homo sapiens (Human))
Oged

US Patent
LigandPNGBDBM362839((R)-(4-fluorophenyl)(8- methyl-3-(5-methylfuran-2-...)
Affinity DataKi:  48nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeuromedin-K receptor(Homo sapiens (Human))
Oged

US Patent
LigandPNGBDBM362839((R)-(4-fluorophenyl)(8- methyl-3-(5-methylfuran-2-...)
Affinity DataIC50:  60nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent