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Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-3' and Ligand = 'BDBM50275306'
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50275306(3-((1H-Pyrrole-1-carbonyloxy)-1-methylpropyl)dimet...)
Affinity DataKi:  100nMAssay Description:Agonist activity at rat alpha-3-beta-4 nAChR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50275306(3-((1H-Pyrrole-1-carbonyloxy)-1-methylpropyl)dimet...)
Affinity DataKi:  1.00E+5nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha-3-beta-4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed