Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Nischarin' and Ligand = 'BDBM50127584'
TargetNischarin(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50127584(6-Chloro-2-(4,5-dihydro-1H-imidazol-2-yl)-4-methyl...)
Affinity DataKi:  140nMAssay Description:In vitro binding affinity determined against imidazoline receptor I-1 from rabbit kidney preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50127584(6-Chloro-2-(4,5-dihydro-1H-imidazol-2-yl)-4-methyl...)
Affinity DataKi:  158nMAssay Description:Binding affinity for imidazoline receptor I-2 in rabbit kidney homogenate (relative to [3H]-Idazoxan radioligand)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50127584(6-Chloro-2-(4,5-dihydro-1H-imidazol-2-yl)-4-methyl...)
Affinity DataKi:  173nMAssay Description:In vitro binding affinity determined against imidazoline receptor I-2 using rabbit kidney preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed