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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50105932'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105932(CHEMBL3598050)
Affinity DataIC50:  15nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105932(CHEMBL3598050)
Affinity DataEC50:  49nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed