Found 1 Enz. Inhib. hit(s) with Target = 'Nuclear receptor corepressor 1' and Ligand = 'BDBM50525179'
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Beijing University Of Chemical Technology
Curated by ChEMBL
Beijing University Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 215nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair