Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group D member 1' and Ligand = 'BDBM50434037'
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50434037(CHEMBL2381208)
Affinity DataEC50:  200nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50434037(CHEMBL2381208)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed