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Found 1 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 3' and Ligand = 'BDBM50146171'
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50146171(CHEMBL3763399)
Affinity DataIC50:  14nMAssay Description:Inverse agonist activity at GST tagged-human CAR-LBD assessed as reduction in fluorescein-PGC1 alpha coactivator recruitment after 1 hr by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed