Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 4 group A member 2' and Ligand = 'BDBM50517851'
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM50517851(CHEMBL4440924)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 2(Mus musculus)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50517851(CHEMBL4440924)
Affinity DataEC50:  1nMAssay Description:Agonist activity at Nurr1 in mouse N2A cells harboring NBRE by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed