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Found 4 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 1' and Ligand = 'BDBM50267999'
TargetP2Y purinoceptor 1(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50267999(({[({[(2R,3S,4R,5R)-5-[6-amino-2-(methylsulfanyl)-...)
Affinity DataEC50:  2.60nMAssay Description:Agonists activity was evaluated by release of [Ca2+] release of HEK 293 cells stably transfected with rat-brain P2Y purinoceptor 1 (P2Y1-R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50267999(({[({[(2R,3S,4R,5R)-5-[6-amino-2-(methylsulfanyl)-...)
Affinity DataEC50:  28nMAssay Description:Agonist activity at rat pancreas P2Y1 receptor assessed as enhancement of insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50267999(({[({[(2R,3S,4R,5R)-5-[6-amino-2-(methylsulfanyl)-...)
Affinity DataEC50:  2.60nMAssay Description:Concentration required for calcium mobilization at rat purinergic 2Y1 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50267999(({[({[(2R,3S,4R,5R)-5-[6-amino-2-(methylsulfanyl)-...)
Affinity DataEC50:  2.60nMAssay Description:Concentration required for calcium mobilization at rat purinergic 2Y1 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed