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Found 2 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform' and Ligand = 'BDBM50137851'
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137851(CHEMBL3752866)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137851(CHEMBL3752866)
Affinity DataIC50:  7.22E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed