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Found 2 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM139677'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM139677(US8894989, 59 | US8894989, 63)
Affinity DataIC50:  19nMpH: 8.0Assay Description:A convenient method to determine IC50 of a PARP inhibitor compound is a PARP assay using purified recombinant human PARP from Trevigan (Gaithersburg,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM139677(US8894989, 59 | US8894989, 63)
Affinity DataIC50:  23nMpH: 8.0Assay Description:A convenient method to determine IC50 of a PARP inhibitor compound is a PARP assay using purified recombinant human PARP from Trevigan (Gaithersburg,...More data for this Ligand-Target Pair
In DepthDetails US Patent