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Found 1 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50120718'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120718(2-Pyridin-3-yl-1,3,4,5-tetrahydro-azepino[5,4,3-cd...)
Affinity DataKi:  7nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed