Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50251657'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50251657(2-(2-(methylamino)propan-2-yl)-1H-benzo[d]imidazol...)
Affinity DataKi:  4nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50251657(2-(2-(methylamino)propan-2-yl)-1H-benzo[d]imidazol...)
Affinity DataEC50:  1.30nMAssay Description:Inhibition of PARP1 (unknown origin) in cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed