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Found 3 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50072018'
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072018(5,8-difluoro-2,2,4-trimethyl-2,10-dihydro-1H-inden...)
Affinity DataKi:  1.5nMAssay Description:Antagonist activity against human progesterone receptor B (hPR-B) in cotransfected CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072018(5,8-difluoro-2,2,4-trimethyl-2,10-dihydro-1H-inden...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]progesterone from Progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072018(5,8-difluoro-2,2,4-trimethyl-2,10-dihydro-1H-inden...)
Affinity DataEC50:  650nMAssay Description:Agonistic activity against human progesterone receptor B (hPR-B) in cotransfected CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed