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Found 8 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50243394'
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50243394((+)-(S)-7,9-difluoro-2,2,4-trimethyl-5-((S)-3-meth...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity at human progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50243394((+)-(S)-7,9-difluoro-2,2,4-trimethyl-5-((S)-3-meth...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity at human progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50243394((+)-(S)-7,9-difluoro-2,2,4-trimethyl-5-((S)-3-meth...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50243394((+)-(S)-7,9-difluoro-2,2,4-trimethyl-5-((S)-3-meth...)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50243394((+)-(S)-7,9-difluoro-2,2,4-trimethyl-5-((S)-3-meth...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50243394((+)-(S)-7,9-difluoro-2,2,4-trimethyl-5-((S)-3-meth...)
Affinity DataEC50:  50.8nMAssay Description:Agonist activity at human progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50243394((+)-(S)-7,9-difluoro-2,2,4-trimethyl-5-((S)-3-meth...)
Affinity DataEC50:  50.8nMAssay Description:Agonist activity at human progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50243394((+)-(S)-7,9-difluoro-2,2,4-trimethyl-5-((S)-3-meth...)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed