Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50375444'
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375444(CHEMBL258861)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivation relative to Org 31710More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed