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Found 2 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 2' and Ligand = 'BDBM50339244'
TargetProteinase-activated receptor 2(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50339244(2-amino-N-((4S,7S,13S,16S)-13-sec-butyl-4-carbamoy...)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at PAR2 in human 16HBE14o cells assessed as increase in intracellular calcium levels by in vitro physiological response assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50339244(2-amino-N-((4S,7S,13S,16S)-13-sec-butyl-4-carbamoy...)
Affinity DataEC50:  142nMAssay Description:Agonist activity at PAR2 in human 16HBE14o cells assessed as increase in intracellular calcium levels measured every 15 second for 2 hrs by xCelligen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed