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Found 3 Enz. Inhib. hit(s) with Target = 'Proto-oncogene tyrosine-protein kinase Src' and Ligand = 'BDBM340069'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM340069((S,E)-4-(8-amino-3-(1-(4- methoxybut-2-enoyl)piper...)
Affinity DataEC50: >1.00E+3nMAssay Description:Src enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Src enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM340069((S,E)-4-(8-amino-3-(1-(4- methoxybut-2-enoyl)piper...)
Affinity DataEC50: >1.00E+3nMAssay Description:Src enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Src enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM340069((S,E)-4-(8-amino-3-(1-(4- methoxybut-2-enoyl)piper...)
Affinity DataEC50: >1.00E+3nMAssay Description:Src enzyme (Millipore catalog #14-326), is diluted to 0.8 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent