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Found 2 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM15168'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM15168(1-{1-[(4-{7-phenyl-1H-pyrazolo[3,4-g]quinoxalin-6-...)
Affinity DataIC50:  85nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM15168(1-{1-[(4-{7-phenyl-1H-pyrazolo[3,4-g]quinoxalin-6-...)
Affinity DataIC50:  85nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt1, Akt2, and Akt3 proteins were monitored for kinase activity in the presence or absence of Akt inhibitors in a 96-well...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed