Found 1 Enz. Inhib. hit(s) with Target = 'Receptor tyrosine-protein kinase erbB-2' and Ligand = 'BDBM297481'
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Madrigal Pharmaceuticals
US Patent
Madrigal Pharmaceuticals
US Patent
Affinity DataIC50: 710nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair