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Found 2 Enz. Inhib. hit(s) with Target = 'Receptor tyrosine-protein kinase erbB-2' and Ligand = 'BDBM332537'
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Arromax Pharmatech

Curated by ChEMBL
LigandPNGBDBM332537((R,E)-N-(4-(3-chloro-4-fluorophenylamino)-7-(2-met...)
Affinity DataIC50:  148nMAssay Description:Inhibition of recombinant human His-tagged HER2 catalytic domain (676 to 1255 residues) expressed in baculovirus expression system using TK-biotin pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Arromax Pharmatech

Curated by ChEMBL
LigandPNGBDBM332537((R,E)-N-(4-(3-chloro-4-fluorophenylamino)-7-(2-met...)
Affinity DataIC50:  148nMAssay Description:The kinase analysis in vitro was performed using the HTRF kinEASE TK kit of Invitrogen Co., the procedure steps were carried out according to instruc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent