Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50053093'
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50053093((2E,4E,6E)-8-Cyclohex-2-en-(E)-ylidene-3,7-dimethy...)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to mouse Retinoic acid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50053093((2E,4E,6E)-8-Cyclohex-2-en-(E)-ylidene-3,7-dimethy...)
Affinity DataKd: >200nMAssay Description:Inhibition of binding to human Retinoic acid receptor RXR DEF domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed