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Found 2 Enz. Inhib. hit(s) with Target = 'Retinol-binding protein 4' and Ligand = 'BDBM50026254'
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026254(CHEMBL3359015)
Affinity DataIC50:  0.481nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026254(CHEMBL3359015)
Affinity DataIC50:  149nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed