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Found 2 Enz. Inhib. hit(s) with Target = 'Segment polarity protein dishevelled homolog DVL-1' and Ligand = 'BDBM50177707'
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177707(CHEMBL3814506)
Affinity DataKd:  1.52E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177707(CHEMBL3814506)
Affinity DataKd:  3.80nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed