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Found 5 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk1' and Ligand = 'BDBM50216165'
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50:  81nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50:  81nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50:  250nMAssay Description:Inhibition of Chk1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed