Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase TBK1' and Ligand = 'BDBM357895'
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM357895(US10214536, Compound 78)
Affinity DataIC50:  750nMAssay Description:Inhibition of human TBK1 (1 to 657 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in presence o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM357895(US10214536, Compound 78)
Affinity DataIC50:  790nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent