Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-1' and Ligand = 'BDBM2683'
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against PIM1More data for this Ligand-Target Pair
Affinity DataIC50: 150nMpH: 7.6 T: 2°CAssay Description:A coupled-enzyme assay was used to quantify the ADP generated in the kinase reaction with S6 peptide (RRRLSSLRA) as the phosphoacceptorsubstrate.More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity to non phosphorylated PIM1More data for this Ligand-Target Pair