Found 9 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50021226'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:Displacement of [125I]RTI-55 from serotonin transporter of frozen rat caudate membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Reuptake inhibitory activity against Serotonin transporterMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 0.440nMAssay Description:Inhibition of dopamine uptake in rat synaptosomal fractionMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 0.480nMAssay Description:Inhibition of 5-HT uptake in rat synaptosomal fractionMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:Inhibition of 5-HT uptake in rat synaptosomal fractionMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals
Curated by PDSP Ki Database
Boots Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:Inhibition of 5-HT uptake in rat synaptosomal fractionMore data for this Ligand-Target Pair