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Found 2 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50275829'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50275829(CHEMBL472253 | N-Ethyl-N-propargyl (1R,2R)-2-(Amin...)
Affinity DataIC50:  81nMAssay Description:Displacement of [alpha,beta-3H(N)]-5-hydroxytryptamine from human cloned SERT expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50275829(CHEMBL472253 | N-Ethyl-N-propargyl (1R,2R)-2-(Amin...)
Affinity DataIC50:  160nMAssay Description:Displacement of [alpha,beta-3H(N)]-5-hydroxytryptamine from rat synaptosomal SERT expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed