Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Solute carrier family 15 member 2' and Ligand = 'BDBM84007'
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Biozentrum Of The Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM84007(CEFIXIME | Cefiximum [Latin] | MLS002222332 | SMR0...)
Affinity DataKi:  2.60E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (pH6.0) in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM84007(CEFIXIME | Cefiximum [Latin] | MLS002222332 | SMR0...)
Affinity DataKi:  2.60E+6nMAssay Description:Binding affinity to human PepT2 in SKTP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Rattus norvegicus)
Biozentrum Of The Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM84007(CEFIXIME | Cefiximum [Latin] | MLS002222332 | SMR0...)
Affinity DataKi:  1.19E+7nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Biozentrum Of The Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM84007(CEFIXIME | Cefiximum [Latin] | MLS002222332 | SMR0...)
Affinity DataIC50:  3.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed