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Found 1 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 3' and Ligand = 'BDBM50053620'
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50053620(1-phenylguanidine | 1N-amino(immino)methylaniline ...)
Affinity DataIC50:  9.98E+4nMAssay Description:Inhibition of human OCT3 expressed in HEK293 cells assessed as decrease in uptake of substrate [3H]MPP+ after 1 min by liquid scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed