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Found 1 Enz. Inhib. hit(s) with Target = 'Solute carrier organic anion transporter family member 2B1' and Ligand = 'BDBM50061554'
TargetSolute carrier organic anion transporter family member 2B1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50061554((+)-Silychristin | (2R,3R)-3,5,7-Trihydroxy-2-[(2R...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of OATP2B1 (unknown origin) expressed in MDCK2 cells assessed as reduction of [3H]estrone-3-sulfate uptake after 3 mins by beta-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed