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Found 2 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 2' and Ligand = 'BDBM50341570'
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50341570(7-Chloro-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperid...)
Affinity DataKi:  0.110nMAssay Description:Displacement of I125-somatostatin-14 from human SST2 expressed in CHO cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50341570(7-Chloro-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperid...)
Affinity DataIC50:  20nMAssay Description:Agonist activity at human SST2 expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP release after 40 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed