Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Stromelysin-1' and Ligand = 'BDBM13086'
TargetStromelysin-1(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM13086(2-[(4-aminobenzene)(2-methylpropyl)sulfonamido]-N-...)
Affinity DataKi:  5.00E+3nM ΔG°:  -31.5kJ/molepH: 7.5 T: 2°CAssay Description:Stromelysin inhibitory activity is based on the hydrolysis of substance P by recombinant human stromelysin to generate a fragment, substance P 7-11, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM13086(2-[(4-aminobenzene)(2-methylpropyl)sulfonamido]-N-...)
Affinity DataKi:  5.01E+3nMAssay Description:Inhibition of human recombinant MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed