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Found 2 Enz. Inhib. hit(s) with Target = 'TGF-beta receptor type-1' and Ligand = 'BDBM282844'
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Syngene International

US Patent
LigandPNGBDBM282844(6-(4-(3-chloro-4-fluorophenyl)-1-isopropyl-1H- imi...)
Affinity DataIC50:  0.600nMAssay Description:Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Syngene International

US Patent
LigandPNGBDBM282844(6-(4-(3-chloro-4-fluorophenyl)-1-isopropyl-1H- imi...)
Affinity DataIC50:  0.600nMpH: 7.4 T: 2°CAssay Description:Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent