Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'Thymidine kinase, cytosolic' and Ligand = 'BDBM50404860'
TargetThymidine kinase, cytosolic(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  1.10E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  2.40E+4nMAssay Description:Competitive inhibition of thymidine kinase in mouse Ehrlich's ascites cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  2.40E+4nMAssay Description:Competitive inhibition of thymidine kinase in mouse Ehrlich's ascites cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Cricetulus griseus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  3.10E+5nMAssay Description:Competitive inhibition of thymidine kinase in BHK21 (C13) cells using thymidine as substrate assessed as formation of TMP by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Cricetulus griseus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  3.10E+5nMAssay Description:Competitive inhibition of thymidine kinase in BHK21 (C13) cells using thymidine as substrate assessed as formation of TMP by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed