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Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50055267'
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50055267(CHEMBL3323682)
Affinity DataIC50:  2.39E+4nMAssay Description:Antagonist activity against human recombinant TRPV1 expressed in HEK293 cells assessed as reduction in capsaicin-induced intracellular calcium respon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50055267(CHEMBL3323682)
Affinity DataEC50:  6.90E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed