Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50055267'
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.39E+4nMAssay Description:Antagonist activity against human recombinant TRPV1 expressed in HEK293 cells assessed as reduction in capsaicin-induced intracellular calcium respon...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataEC50: 6.90E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluorescence assayMore data for this Ligand-Target Pair