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Found 4 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50440401'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50440401(CHEMBL2425550)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50440401(CHEMBL2425550)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]RTX from human TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50440401(CHEMBL2425550)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50440401(CHEMBL2425550)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed