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Found
1
Enz. Inhib. hit(s) with Target = 'Tryptophan 2,3-dioxygenase' and Ligand = 'BDBM339929'
Target
Tryptophan 2,3-dioxygenase
(Homo sapiens (Human))
Iteos Therapeutics
US Patent
Ligand
BDBM339929
(6-fluoro-3-(6-(piperidin-4- yloxy)pyridin-3-yl)-1H...)
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Affinity Data
IC50: 560nM
Assay Description:
The compounds of formula I inhibit the enzymatic activity of human TDO2.To measure the TDO2 activity, the procedure described in Dolusic et al. J. Me...
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Target Info
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Ligand Info
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US Patent
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