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Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1' and Ligand = 'BDBM50244527'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50244527(9-(2-(1H-indazol-4-yl)vinyl)-N-(4-(dimethylphospho...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of Abl kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50244527(9-(2-(1H-indazol-4-yl)vinyl)-N-(4-(dimethylphospho...)
Affinity DataIC50:  2.40nMAssay Description:In vitro kinase assay using Abl, Abl T315I or Src kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed