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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK' and Ligand = 'BDBM50457319'
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50457319(CHEMBL4205974 | US10662187, Compound 59 | US107935...)
Affinity DataIC50:  10nMAssay Description:Inhibition of BTK (unknown origin) using peptide substrate after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50457319(CHEMBL4205974 | US10662187, Compound 59 | US107935...)
Affinity DataIC50:  55nMAssay Description:Btk kinase activity was determined using a homogenous time resolved fluorescence (HTRF) methodology. Measurements were performed in a reaction volume...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50457319(CHEMBL4205974 | US10662187, Compound 59 | US107935...)
Affinity DataIC50:  55nMAssay Description:Measurements were performed in a reaction volume of 15 μL using 384-well assay plates. Kinase enzyme, inhibitor, ATP and 1 μM peptide subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent