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Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ITK/TSK' and Ligand = 'BDBM191628'
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Pharmacyclics

US Patent
LigandPNGBDBM191628(US9181263, 24 | US9278100, 24)
Affinity DataIC50:  476nMAssay Description:IC50s were determined using the in vitro HotSpot kinase assay (purified enzymes, 33P-ATP, an appropriate substrate and 1 uM ATP.). Reaction condition...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Pharmacyclics

US Patent
LigandPNGBDBM191628(US9181263, 24 | US9278100, 24)
Affinity DataIC50:  476nMAssay Description:IC50s were determined using the in vitro HotSpot kinase assay (purified enzymes, 33P-ATP, an appropriate substrate and 1 μM ATP.). For enzyme in...More data for this Ligand-Target Pair
In DepthDetails US Patent