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Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK2' and Ligand = 'BDBM409858'
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Hutchison Medipharma

US Patent
LigandPNGBDBM409858((R)—N-(1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyr...)
Affinity DataIC50: <100nMAssay Description:JAK1/2/3 kinase assay are performed in vitro using Kit-Tyr 6 Peptide (Invitrogen, Cat. No. PV4122). TYK2 kinase assay are performed in vitro using Z&...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent