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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Uracil nucleotide/cysteinyl leukotriene receptor' and Ligand = 'BDBM50010475'   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Uracil nucleotide/cysteinyl leukotriene receptor


(Homo sapiens)
BDBM50010475
PNG
(GAVESTINEL | GV-150526X)
Show SMILES OC(=O)c1[nH]c2cc(Cl)cc(Cl)c2c1\C=C\C(=O)Nc1ccccc1
Show InChI InChI=1S/C18H12Cl2N2O3/c19-10-8-13(20)16-12(17(18(24)25)22-14(16)9-10)6-7-15(23)21-11-4-2-1-3-5-11/h1-9,22H,(H,21,23)(H,24,25)/b7-6+
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KEGG

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PC cid
PC sid
UniChem
AffyNet 
Article
1.63E+3n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]PSB-12150 from human GPR17 expressed in CHO-K1 cell membranes after 60 mins by heterologous competition binding assay


Citation and Details
More data for this
Ligand-Target Pair