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Found 2 Enz. Inhib. hit(s) with Target = 'Vascular endothelial growth factor receptor 2' and Ligand = 'BDBM5328'
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM5328(2-quinolinone deriv. 3 | 3-(1H-indol-2-yl)-1,2-dih...)
Affinity DataIC50:  8nMAssay Description:Inhibition of VEGFR-2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM5328(2-quinolinone deriv. 3 | 3-(1H-indol-2-yl)-1,2-dih...)
Affinity DataIC50:  8nMpH: 7.4 T: 2°CAssay Description:Activated KDR was incubated with 25 uM/10 uCi of [gamma-33P] ATP, poly-Glu/Tyr, and inhibitors in kinase buffer for 15 min at 22 °C. The reactio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed