Affinity DataKi: 0.234nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.234nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 21.9nMAssay Description:Displacement of [3H]AVP from rat V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 21.9nMAssay Description:Displacement of [3H]AVP from rat V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 55.0nMAssay Description:Antagonist activity at human V1A receptor expressed in CHO cells assessed as inhibition of AVP-induced intracellular calcium releaseMore data for this Ligand-Target Pair