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Compile Data Set for Download or QSAR

Found 26 hits of Enz. Inhib. data with enzyme = 'Adenosine receptor A2a' and Substrate = 'to-be-curated'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM415451
PNG
(3-Ethyl-1-(2-methoxyethyl)-5-methyl-6-[(2-oxo-2,3-...)
Show SMILES CCn1c(=O)n(CCOC)c2sc(Cn3cc[nH]c3=O)c(C)c2c1=O
Show InChI InChI=1S/C16H20N4O4S/c1-4-19-13(21)12-10(2)11(9-18-6-5-17-15(18)22)25-14(12)20(16(19)23)7-8-24-3/h5-6H,4,7-9H2,1-3H3,(H,17,22)
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100n/an/an/an/an/an/an/an/a



BAYER PHARMA AKTIENGESELLSCHAFT

US Patent


Assay Description
The binding properties of the test compounds on adenosine receptors were determined in binding studies with radioligands. For this purpose, membrane ...


US Patent US10428083 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM415448
PNG
(3-Ethyl-1-(2-methoxyethyl)-5-methyl-6-[(2-oxoimida...)
Show SMILES CCn1c(=O)n(CCOC)c2sc(CN3CCNC3=O)c(C)c2c1=O
Show InChI InChI=1S/C16H22N4O4S/c1-4-19-13(21)12-10(2)11(9-18-6-5-17-15(18)22)25-14(12)20(16(19)23)7-8-24-3/h4-9H2,1-3H3,(H,17,22)
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120n/an/an/an/an/an/an/an/a



BAYER PHARMA AKTIENGESELLSCHAFT

US Patent


Assay Description
The binding properties of the test compounds on adenosine receptors were determined in binding studies with radioligands. For this purpose, membrane ...


US Patent US10428083 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM415450
PNG
(3-Isopropyl-1-(2-methoxyethyl)-5-methyl-6-[(2-oxoi...)
Show SMILES COCCn1c2sc(CN3CCNC3=O)c(C)c2c(=O)n(C(C)C)c1=O
Show InChI InChI=1S/C17H24N4O4S/c1-10(2)21-14(22)13-11(3)12(9-19-6-5-18-16(19)23)26-15(13)20(17(21)24)7-8-25-4/h10H,5-9H2,1-4H3,(H,18,23)
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270n/an/an/an/an/an/an/an/a



BAYER PHARMA AKTIENGESELLSCHAFT

US Patent


Assay Description
The binding properties of the test compounds on adenosine receptors were determined in binding studies with radioligands. For this purpose, membrane ...


US Patent US10428083 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM415449
PNG
(3-Ethyl-5-methyl-1-(oxetan-2-ylmethyl)-6-[(2-oxoim...)
Show SMILES CCn1c(=O)n(CC2CCO2)c2sc(CN3CCNC3=O)c(C)c2c1=O
Show InChI InChI=1S/C17H22N4O4S/c1-3-20-14(22)13-10(2)12(9-19-6-5-18-16(19)23)26-15(13)21(17(20)24)8-11-4-7-25-11/h11H,3-9H2,1-2H3,(H,18,23)
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280n/an/an/an/an/an/an/an/a



BAYER PHARMA AKTIENGESELLSCHAFT

US Patent


Assay Description
The binding properties of the test compounds on adenosine receptors were determined in binding studies with radioligands. For this purpose, membrane ...


US Patent US10428083 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375228
PNG
(3-bromo-6-(pyridin-3-yl)-5-(pyridin-4-yl)pyridin-2...)
Show SMILES Nc1cc(Br)c(-c2ccncc2)c(n1)-c1cccnc1
Show InChI InChI=1S/C15H11BrN4/c16-12-8-13(17)20-15(11-2-1-5-19-9-11)14(12)10-3-6-18-7-4-10/h1-9H,(H2,17,20)
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300n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375227
PNG
(3-chloro-6-(pyridin-3-yl)-5-(pyridin-4-yl)pyridin-...)
Show SMILES Nc1cc(Cl)c(-c2ccncc2)c(n1)-c1cccnc1
Show InChI InChI=1S/C15H11ClN4/c16-12-8-13(17)20-15(11-2-1-5-19-9-11)14(12)10-3-6-18-7-4-10/h1-9H,(H2,17,20)
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500n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377143
PNG
((1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethy...)
Show SMILES Nc1nc(nc2n(cnc12)C1O[C@H](CO)[C@@H](O)[C@H]1O)-n1cc(cn1)C(=O)NC1CCCC1
Show InChI InChI=1/C19H24N8O5/c20-15-12-16(26(8-21-12)18-14(30)13(29)11(7-28)32-18)25-19(24-15)27-6-9(5-22-27)17(31)23-10-3-1-2-4-10/h5-6,8,10-11,13-14,18,28-30H,1-4,7H2,(H,23,31)(H2,20,24,25)/t11-,13-,14-,18?/s2
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505n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377141
PNG
((1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydrozymethy...)
Show SMILES CCNC(=O)c1cnn(c1)-c1nc(N)c2ncn(C3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
Show InChI InChI=1/C16H20N8O5/c1-2-18-14(28)7-3-20-24(4-7)16-21-12(17)9-13(22-16)23(6-19-9)15-11(27)10(26)8(5-25)29-15/h3-4,6,8,10-11,15,25-27H,2,5H2,1H3,(H,18,28)(H2,17,21,22)/t8-,10-,11-,15?/s2
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505n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377140
PNG
((1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethy...)
Show SMILES CN(C)C(=O)c1cnn(c1)-c1nc(N)c2ncn(C3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
Show InChI InChI=1/C16H20N8O5/c1-22(2)14(28)7-3-19-24(4-7)16-20-12(17)9-13(21-16)23(6-18-9)15-11(27)10(26)8(5-25)29-15/h3-4,6,8,10-11,15,25-27H,5H2,1-2H3,(H2,17,20,21)/t8-,10-,11-,15?/s2
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505n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377142
PNG
(1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Show SMILES NC(=O)c1cnn(c1)-c1nc(N)c2ncn(C3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
Show InChI InChI=1/C14H16N8O5/c15-10-7-12(20-14(19-10)22-2-5(1-18-22)11(16)26)21(4-17-7)13-9(25)8(24)6(3-23)27-13/h1-2,4,6,8-9,13,23-25H,3H2,(H2,16,26)(H2,15,19,20)/t6-,8-,9-,13?/s2
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505n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377134
PNG
(Ethyl 1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxy...)
Show SMILES CCOC(=O)c1cnn(c1)-c1nc(N)c2ncn(C3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
Show InChI InChI=1/C16H19N7O6/c1-2-28-15(27)7-3-19-23(4-7)16-20-12(17)9-13(21-16)22(6-18-9)14-11(26)10(25)8(5-24)29-14/h3-4,6,8,10-11,14,24-26H,2,5H2,1H3,(H2,17,20,21)/t8-,10-,11-,14?/s2
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505n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377144
PNG
((1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethy...)
Show SMILES Nc1nc(nc2n(cnc12)C1O[C@H](CO)[C@@H](O)[C@H]1O)-n1cc(cn1)C(=O)NCc1ccc(Cl)cc1
Show InChI InChI=1/C21H21ClN8O5/c22-12-3-1-10(2-4-12)5-24-19(34)11-6-26-30(7-11)21-27-17(23)14-18(28-21)29(9-25-14)20-16(33)15(32)13(8-31)35-20/h1-4,6-7,9,13,15-16,20,31-33H,5,8H2,(H,24,34)(H2,23,27,28)/t13-,15-,16-,20?/s2
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505n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375232
PNG
(3-chloro-5-(3-fluoropyridin-4-yl)-6-(pyridin-4-yl)...)
Show SMILES Nc1cc(Cl)c(-c2ccnc(F)c2)c(n1)-c1ccncc1
Show InChI InChI=1S/C15H10ClFN4/c16-11-8-13(18)21-15(9-1-4-19-5-2-9)14(11)10-3-6-20-12(17)7-10/h1-8H,(H2,18,21)
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555n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM415453
PNG
(3-Ethyl-5-methyl-6-[(5-oxo-1,5-dihydro-4H-1,2,4-tr...)
Show SMILES CCn1c(=O)n(CCC(F)(F)F)c2sc(Cn3cn[nH]c3=O)c(C)c2c1=O
Show InChI InChI=1S/C15H16F3N5O3S/c1-3-22-11(24)10-8(2)9(6-21-7-19-20-13(21)25)27-12(10)23(14(22)26)5-4-15(16,17)18/h7H,3-6H2,1-2H3,(H,20,25)
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790n/an/an/an/an/an/an/an/a



BAYER PHARMA AKTIENGESELLSCHAFT

US Patent


Assay Description
The binding properties of the test compounds on adenosine receptors were determined in binding studies with radioligands. For this purpose, membrane ...


US Patent US10428083 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377139
PNG
(1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Show SMILES Nc1nc(nc2n(cnc12)C1O[C@H](CO)[C@@H](O)[C@H]1O)-n1cc(cn1)C(O)=O
Show InChI InChI=1/C14H15N7O6/c15-10-7-11(19-14(18-10)21-2-5(1-17-21)13(25)26)20(4-16-7)12-9(24)8(23)6(3-22)27-12/h1-2,4,6,8-9,12,22-24H,3H2,(H,25,26)(H2,15,18,19)/t6-,8-,9-,12?/s2
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>1.00E+3n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375233
PNG
(3-bromo-5-(3-fluoropyridin-4-yl)-6-(pyridin-4-yl)p...)
Show SMILES Nc1cc(Br)c(-c2ccnc(F)c2)c(n1)-c1ccncc1
Show InChI InChI=1S/C15H10BrFN4/c16-11-8-13(18)21-15(9-1-4-19-5-2-9)14(11)10-3-6-20-12(17)7-10/h1-8H,(H2,18,21)
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1.30E+3n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM415452
PNG
(3-Ethyl-5-methyl-6-[(5-oxo-4,5-dihydro-1H-1,2,4-tr...)
Show SMILES CCn1c(=O)n(CCC(F)(F)F)c2sc(Cn3nc[nH]c3=O)c(C)c2c1=O
Show InChI InChI=1S/C15H16F3N5O3S/c1-3-21-11(24)10-8(2)9(6-23-13(25)19-7-20-23)27-12(10)22(14(21)26)5-4-15(16,17)18/h7H,3-6H2,1-2H3,(H,19,20,25)
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1.70E+3n/an/an/an/an/an/an/an/a



BAYER PHARMA AKTIENGESELLSCHAFT

US Patent


Assay Description
The binding properties of the test compounds on adenosine receptors were determined in binding studies with radioligands. For this purpose, membrane ...


US Patent US10428083 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375229
PNG
(3-chloro-5-(3-fluoropyridin-4-yl)-6-(pyridin-3-yl)...)
Show SMILES Nc1cc(Cl)c(-c2ccnc(F)c2)c(n1)-c1cccnc1
Show InChI InChI=1S/C15H10ClFN4/c16-11-7-13(18)21-15(10-2-1-4-19-8-10)14(11)9-3-5-20-12(17)6-9/h1-8H,(H2,18,21)
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4.80E+3n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375231
PNG
(3-chloro-6-(5-fluoropyridin-3-yl)-5-(3-fluoropyrid...)
Show SMILES Nc1cc(Cl)c(-c2ccnc(F)c2)c(n1)-c1cncc(F)c1
Show InChI InChI=1S/C15H9ClF2N4/c16-11-5-13(19)22-15(9-3-10(17)7-20-6-9)14(11)8-1-2-21-12(18)4-8/h1-7H,(H2,19,22)
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>5.00E+3n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375226
PNG
(5-(3-fluoropyridin-4-yl)-6-(pyridin-4-yl)pyridin-2...)
Show SMILES Nc1ccc(-c2ccnc(F)c2)c(n1)-c1ccncc1
Show InChI InChI=1S/C15H11FN4/c16-13-9-11(5-8-19-13)12-1-2-14(17)20-15(12)10-3-6-18-7-4-10/h1-9H,(H2,17,20)
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>5.00E+3n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375230
PNG
(3-bromo-5-(3-fluoropyridin-4-yl)-6-(pyridin-3-yl)p...)
Show SMILES Nc1cc(Br)c(-c2ccnc(F)c2)c(n1)-c1cccnc1
Show InChI InChI=1S/C15H10BrFN4/c16-11-7-13(18)21-15(10-2-1-4-19-8-10)14(11)9-3-5-20-12(17)6-9/h1-8H,(H2,18,21)
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>5.00E+3n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(Homo sapiens (Human))
BDBM375234
PNG
(3-chloro-5-(3-fluoropyridin-4-yl)-6-(6-methoxypyri...)
Show SMILES COc1ccc(cn1)-c1nc(N)cc(Cl)c1-c1ccnc(F)c1
Show InChI InChI=1S/C16H12ClFN4O/c1-23-14-3-2-10(8-21-14)16-15(11(17)7-13(19)22-16)9-4-5-20-12(18)6-9/h2-8H,1H3,(H2,19,22)
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>5.00E+3n/an/an/an/an/an/an/an/a



Palobiofarma, S.L.

US Patent


Assay Description
The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...


US Patent US10253017 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM50152084
PNG
(1-[6-Amino-9-(3,4-dihydroxy-5-hydroxymethyl-tetrah...)
Show SMILES CNC(=O)c1cnn(c1)-c1nc(N)c2ncn(C3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
Show InChI InChI=1S/C15H18N8O5/c1-17-13(27)6-2-19-23(3-6)15-20-11(16)8-12(21-15)22(5-18-8)14-10(26)9(25)7(4-24)28-14/h2-3,5,7,9-10,14,24-26H,4H2,1H3,(H,17,27)(H2,16,20,21)/t7-,9-,10-,14?/m1/s1
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US Patent
5.50E+3n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377137
PNG
((4S,2R,3R,5R)-2-{6-Amino2-[4-(4-methylphenyl)pyraz...)
Show SMILES Cc1ccc(cc1)-c1cnn(c1)-c1nc(N)c2ncn(C3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
Show InChI InChI=1/C20H21N7O4/c1-10-2-4-11(5-3-10)12-6-23-27(7-12)20-24-17(21)14-18(25-20)26(9-22-14)19-16(30)15(29)13(8-28)31-19/h2-7,9,13,15-16,19,28-30H,8H2,1H3,(H2,21,24,25)/t13-,15-,16-,19?/s2
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5.50E+3n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377135
PNG
((4S,2R,3R,5R)-2-{6-Amino-2-[4-(4-chlorophenyl)pyra...)
Show SMILES Nc1nc(nc2n(cnc12)C1O[C@H](CO)[C@@H](O)[C@H]1O)-n1cc(cn1)-c1ccc(Cl)cc1
Show InChI InChI=1/C19H18ClN7O4/c20-11-3-1-9(2-4-11)10-5-23-27(6-10)19-24-16(21)13-17(25-19)26(8-22-13)18-15(30)14(29)12(7-28)31-18/h1-6,8,12,14-15,18,28-30H,7H2,(H2,21,24,25)/t12-,14-,15-,18?/s2
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5.50E+3n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair
Adenosine receptor A2a


(GUINEA PIG)
BDBM377136
PNG
((4S,2R,3R,5R)-2-{6-Amino-2-[4-(4-metboxyphenyl)pyr...)
Show SMILES Nc1nc(nc2n(cnc12)C1O[C@H](CO)[C@@H](O)[C@H]1O)-n1cc(cn1)-c1ccc(CO)cc1
Show InChI InChI=1/C20H21N7O5/c21-17-14-18(26(9-22-14)19-16(31)15(30)13(8-29)32-19)25-20(24-17)27-6-12(5-23-27)11-3-1-10(7-28)2-4-11/h1-6,9,13,15-16,19,28-31H,7-8H2,(H2,21,24,25)/t13-,15-,16-,19?/s2
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5.50E+3n/an/an/an/an/an/an/an/a



Gilead Sciences Inc

US Patent


Assay Description
Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...


US Patent USRE47351 (2019)

More data for this
Ligand-Target Pair