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Found 54 hits of Enz. Inhib. data with enzyme = 'Collagenase' and Substrate = '5-FAM/QXL520'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Collagenase


(homo sapiens (human))
BDBM28864
PNG
(2-[(5Z)-5-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]me...)
Show SMILES COc1ccc(cc1)-c1cc(\C=C2/SC(=S)N(CC(O)=O)C2=O)no1
Show InChI InChI=1S/C16H12N2O5S2/c1-22-11-4-2-9(3-5-11)12-6-10(17-23-12)7-13-15(21)18(8-14(19)20)16(24)25-13/h2-7H,8H2,1H3,(H,19,20)/b13-7-
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n/an/a 6.62E+3n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28863
PNG
(2-[(5Z)-5-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]met...)
Show SMILES Cc1ccc(cc1)-c1cc(\C=C2/SC(=S)N(CC(O)=O)C2=O)no1
Show InChI InChI=1S/C16H12N2O4S2/c1-9-2-4-10(5-3-9)12-6-11(17-22-12)7-13-15(21)18(8-14(19)20)16(23)24-13/h2-7H,8H2,1H3,(H,19,20)/b13-7-
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n/an/a<1.00E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28866
PNG
(2-[(5Z)-5-{[5-(4-fluorophenyl)-1,2-oxazol-3-yl]met...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccc(F)cc2)C1=O
Show InChI InChI=1S/C15H9FN2O4S2/c16-9-3-1-8(2-4-9)11-5-10(17-22-11)6-12-14(21)18(7-13(19)20)15(23)24-12/h1-6H,7H2,(H,19,20)/b12-6-
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n/an/a 1.00E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28895
PNG
(2-[(5Z)-5-[(2-methylquinolin-6-yl)methylidene]-4-o...)
Show SMILES Cc1ccc2cc(\C=C3/SC(=S)N(CC(O)=O)C3=O)ccc2n1
Show InChI InChI=1S/C16H12N2O3S2/c1-9-2-4-11-6-10(3-5-12(11)17-9)7-13-15(21)18(8-14(19)20)16(22)23-13/h2-7H,8H2,1H3,(H,19,20)/b13-7-
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n/an/a 1.80E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28865
PNG
(2-[(5Z)-5-{[5-(4-chlorophenyl)-1,2-oxazol-3-yl]met...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccc(Cl)cc2)C1=O
Show InChI InChI=1S/C15H9ClN2O4S2/c16-9-3-1-8(2-4-9)11-5-10(17-22-11)6-12-14(21)18(7-13(19)20)15(23)24-12/h1-6H,7H2,(H,19,20)/b12-6-
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n/an/a 1.92E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28903
PNG
(2-{5-[(3Z)-1-{[(3-chlorophenyl)carbamoyl]methyl}-2...)
Show SMILES OC(=O)CN1C(=S)S\C(C1=O)=C1/C(=O)N(CC(=O)Nc2cccc(Cl)c2)c2ccccc12
Show InChI InChI=1S/C21H14ClN3O5S2/c22-11-4-3-5-12(8-11)23-15(26)9-24-14-7-2-1-6-13(14)17(19(24)29)18-20(30)25(10-16(27)28)21(31)32-18/h1-8H,9-10H2,(H,23,26)(H,27,28)/b18-17-
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n/an/a>2.50E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28903
PNG
(2-{5-[(3Z)-1-{[(3-chlorophenyl)carbamoyl]methyl}-2...)
Show SMILES OC(=O)CN1C(=S)S\C(C1=O)=C1/C(=O)N(CC(=O)Nc2cccc(Cl)c2)c2ccccc12
Show InChI InChI=1S/C21H14ClN3O5S2/c22-11-4-3-5-12(8-11)23-15(26)9-24-14-7-2-1-6-13(14)17(19(24)29)18-20(30)25(10-16(27)28)21(31)32-18/h1-8H,9-10H2,(H,23,26)(H,27,28)/b18-17-
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n/an/a>2.50E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28892
PNG
(2-[(5Z)-5-{[4-(4-methyl-1,4-diazepan-1-yl)phenyl]m...)
Show SMILES CN1CCCN(CC1)c1ccc(\C=C2/SC(=S)N(CC(O)=O)C2=O)cc1
Show InChI InChI=1S/C18H21N3O3S2/c1-19-7-2-8-20(10-9-19)14-5-3-13(4-6-14)11-15-17(24)21(12-16(22)23)18(25)26-15/h3-6,11H,2,7-10,12H2,1H3,(H,22,23)/b15-11-
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n/an/a>2.50E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28892
PNG
(2-[(5Z)-5-{[4-(4-methyl-1,4-diazepan-1-yl)phenyl]m...)
Show SMILES CN1CCCN(CC1)c1ccc(\C=C2/SC(=S)N(CC(O)=O)C2=O)cc1
Show InChI InChI=1S/C18H21N3O3S2/c1-19-7-2-8-20(10-9-19)14-5-3-13(4-6-14)11-15-17(24)21(12-16(22)23)18(25)26-15/h3-6,11H,2,7-10,12H2,1H3,(H,22,23)/b15-11-
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n/an/a>2.50E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28867
PNG
(2-[(5Z)-5-{[5-(4-bromophenyl)-1,2-oxazol-3-yl]meth...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccc(Br)cc2)C1=O
Show InChI InChI=1S/C15H9BrN2O4S2/c16-9-3-1-8(2-4-9)11-5-10(17-22-11)6-12-14(21)18(7-13(19)20)15(23)24-12/h1-6H,7H2,(H,19,20)/b12-6-
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n/an/a 2.74E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28861
PNG
(2-[(5Z)-5-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyli...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccco2)C1=O
Show InChI InChI=1S/C13H8N2O5S2/c16-11(17)6-15-12(18)10(22-13(15)21)5-7-4-9(20-14-7)8-2-1-3-19-8/h1-5H,6H2,(H,16,17)/b10-5-
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n/an/a 3.94E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28899
PNG
(2-[(5Z)-5-[(5-bromo-1-benzothiophen-3-yl)methylide...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2csc3ccc(Br)cc23)C1=O
Show InChI InChI=1S/C14H8BrNO3S3/c15-8-1-2-10-9(4-8)7(6-21-10)3-11-13(19)16(5-12(17)18)14(20)22-11/h1-4,6H,5H2,(H,17,18)/b11-3-
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n/an/a 4.69E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28889
PNG
(2-[(5Z)-5-{[5-(morpholin-4-yl)thiophen-2-yl]methyl...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2ccc(s2)N2CCOCC2)C1=O
Show InChI InChI=1S/C14H14N2O4S3/c17-12(18)8-16-13(19)10(23-14(16)21)7-9-1-2-11(22-9)15-3-5-20-6-4-15/h1-2,7H,3-6,8H2,(H,17,18)/b10-7-
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n/an/a 4.71E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28862
PNG
(2-[(5Z)-4-oxo-5-[(5-phenyl-1,2-oxazol-3-yl)methyli...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccccc2)C1=O
Show InChI InChI=1S/C15H10N2O4S2/c18-13(19)8-17-14(20)12(23-15(17)22)7-10-6-11(21-16-10)9-4-2-1-3-5-9/h1-7H,8H2,(H,18,19)/b12-7-
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n/an/a 5.00E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28888
PNG
(2-[(5Z)-5-({7-bromo-2H,3H-thieno[3,4-b][1,4]dioxin...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2sc(Br)c3OCCOc23)C1=O
Show InChI InChI=1S/C12H8BrNO5S3/c13-10-9-8(18-1-2-19-9)5(21-10)3-6-11(17)14(4-7(15)16)12(20)22-6/h3H,1-2,4H2,(H,15,16)/b6-3-
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n/an/a 5.06E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28889
PNG
(2-[(5Z)-5-{[5-(morpholin-4-yl)thiophen-2-yl]methyl...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2ccc(s2)N2CCOCC2)C1=O
Show InChI InChI=1S/C14H14N2O4S3/c17-12(18)8-16-13(19)10(23-14(16)21)7-9-1-2-11(22-9)15-3-5-20-6-4-15/h1-2,7H,3-6,8H2,(H,17,18)/b10-7-
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n/an/a 6.49E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28899
PNG
(2-[(5Z)-5-[(5-bromo-1-benzothiophen-3-yl)methylide...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2csc3ccc(Br)cc23)C1=O
Show InChI InChI=1S/C14H8BrNO3S3/c15-8-1-2-10-9(4-8)7(6-21-10)3-11-13(19)16(5-12(17)18)14(20)22-11/h1-4,6H,5H2,(H,17,18)/b11-3-
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n/an/a 6.49E+4n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28897
PNG
(2-[(5Z)-5-[(6-bromopyridin-2-yl)methylidene]-4-oxo...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cccc(Br)n2)C1=O
Show InChI InChI=1S/C11H7BrN2O3S2/c12-8-3-1-2-6(13-8)4-7-10(17)14(5-9(15)16)11(18)19-7/h1-4H,5H2,(H,15,16)/b7-4-
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n/an/a>1.00E+5n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28902
PNG
(2-[(5Z)-5-[(5-bromo-1H-indol-3-yl)methylidene]-4-o...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2c[nH]c3ccc(Br)cc23)C1=O
Show InChI InChI=1S/C14H9BrN2O3S2/c15-8-1-2-10-9(4-8)7(5-16-10)3-11-13(20)17(6-12(18)19)14(21)22-11/h1-5,16H,6H2,(H,18,19)/b11-3-
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n/an/a>1.00E+5n/an/an/an/an/an/a



Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28900
PNG
(2-[(5Z)-4-oxo-2-sulfanylidene-5-{thieno[2,3-b]pyra...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc3nccnc3s2)C1=O
Show InChI InChI=1S/C12H7N3O3S3/c16-9(17)5-15-11(18)8(21-12(15)19)4-6-3-7-10(20-6)14-2-1-13-7/h1-4H,5H2,(H,16,17)/b8-4-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28901
PNG
(2-[(5Z)-5-(1H-indol-3-ylmethylidene)-4-oxo-2-sulfa...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2c[nH]c3ccccc23)C1=O
Show InChI InChI=1S/C14H10N2O3S2/c17-12(18)7-16-13(19)11(21-14(16)20)5-8-6-15-10-4-2-1-3-9(8)10/h1-6,15H,7H2,(H,17,18)/b11-5-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28858
PNG
(2-[(5Z)-5-[(2,5-dimethyl-1,3-oxazol-4-yl)methylide...)
Show SMILES Cc1nc(\C=C2/SC(=S)N(CC(O)=O)C2=O)c(C)o1
Show InChI InChI=1S/C11H10N2O4S2/c1-5-7(12-6(2)17-5)3-8-10(16)13(4-9(14)15)11(18)19-8/h3H,4H2,1-2H3,(H,14,15)/b8-3-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28859
PNG
(2-[(5Z)-5-[(2-{1-[(tert-butoxy)carbonyl]piperidin-...)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)c1nc(\C=C2/SC(=S)N(CC(O)=O)C2=O)cs1
Show InChI InChI=1S/C19H23N3O5S3/c1-19(2,3)27-17(26)21-6-4-11(5-7-21)15-20-12(10-29-15)8-13-16(25)22(9-14(23)24)18(28)30-13/h8,10-11H,4-7,9H2,1-3H3,(H,23,24)/b13-8-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28860
PNG
(2-[(5Z)-5-[(2-methyl-4-phenyl-1,3-thiazol-5-yl)met...)
Show SMILES Cc1nc(c(\C=C2/SC(=S)N(CC(O)=O)C2=O)s1)-c1ccccc1
Show InChI InChI=1S/C16H12N2O3S3/c1-9-17-14(10-5-3-2-4-6-10)11(23-9)7-12-15(21)18(8-13(19)20)16(22)24-12/h2-7H,8H2,1H3,(H,19,20)/b12-7-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28862
PNG
(2-[(5Z)-4-oxo-5-[(5-phenyl-1,2-oxazol-3-yl)methyli...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccccc2)C1=O
Show InChI InChI=1S/C15H10N2O4S2/c18-13(19)8-17-14(20)12(23-15(17)22)7-10-6-11(21-16-10)9-4-2-1-3-5-9/h1-7H,8H2,(H,18,19)/b12-7-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28867
PNG
(2-[(5Z)-5-{[5-(4-bromophenyl)-1,2-oxazol-3-yl]meth...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccc(Br)cc2)C1=O
Show InChI InChI=1S/C15H9BrN2O4S2/c16-9-3-1-8(2-4-9)11-5-10(17-22-11)6-12-14(21)18(7-13(19)20)15(23)24-12/h1-6H,7H2,(H,19,20)/b12-6-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28858
PNG
(2-[(5Z)-5-[(2,5-dimethyl-1,3-oxazol-4-yl)methylide...)
Show SMILES Cc1nc(\C=C2/SC(=S)N(CC(O)=O)C2=O)c(C)o1
Show InChI InChI=1S/C11H10N2O4S2/c1-5-7(12-6(2)17-5)3-8-10(16)13(4-9(14)15)11(18)19-8/h3H,4H2,1-2H3,(H,14,15)/b8-3-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28859
PNG
(2-[(5Z)-5-[(2-{1-[(tert-butoxy)carbonyl]piperidin-...)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)c1nc(\C=C2/SC(=S)N(CC(O)=O)C2=O)cs1
Show InChI InChI=1S/C19H23N3O5S3/c1-19(2,3)27-17(26)21-6-4-11(5-7-21)15-20-12(10-29-15)8-13-16(25)22(9-14(23)24)18(28)30-13/h8,10-11H,4-7,9H2,1-3H3,(H,23,24)/b13-8-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28860
PNG
(2-[(5Z)-5-[(2-methyl-4-phenyl-1,3-thiazol-5-yl)met...)
Show SMILES Cc1nc(c(\C=C2/SC(=S)N(CC(O)=O)C2=O)s1)-c1ccccc1
Show InChI InChI=1S/C16H12N2O3S3/c1-9-17-14(10-5-3-2-4-6-10)11(23-9)7-12-15(21)18(8-13(19)20)16(22)24-12/h2-7H,8H2,1H3,(H,19,20)/b12-7-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28861
PNG
(2-[(5Z)-5-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyli...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccco2)C1=O
Show InChI InChI=1S/C13H8N2O5S2/c16-11(17)6-15-12(18)10(22-13(15)21)5-7-4-9(20-14-7)8-2-1-3-19-8/h1-5H,6H2,(H,16,17)/b10-5-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28863
PNG
(2-[(5Z)-5-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]met...)
Show SMILES Cc1ccc(cc1)-c1cc(\C=C2/SC(=S)N(CC(O)=O)C2=O)no1
Show InChI InChI=1S/C16H12N2O4S2/c1-9-2-4-10(5-3-9)12-6-11(17-22-12)7-13-15(21)18(8-14(19)20)16(23)24-13/h2-7H,8H2,1H3,(H,19,20)/b13-7-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28864
PNG
(2-[(5Z)-5-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]me...)
Show SMILES COc1ccc(cc1)-c1cc(\C=C2/SC(=S)N(CC(O)=O)C2=O)no1
Show InChI InChI=1S/C16H12N2O5S2/c1-22-11-4-2-9(3-5-11)12-6-10(17-23-12)7-13-15(21)18(8-14(19)20)16(24)25-13/h2-7H,8H2,1H3,(H,19,20)/b13-7-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28865
PNG
(2-[(5Z)-5-{[5-(4-chlorophenyl)-1,2-oxazol-3-yl]met...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccc(Cl)cc2)C1=O
Show InChI InChI=1S/C15H9ClN2O4S2/c16-9-3-1-8(2-4-9)11-5-10(17-22-11)6-12-14(21)18(7-13(19)20)15(23)24-12/h1-6H,7H2,(H,19,20)/b12-6-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28866
PNG
(2-[(5Z)-5-{[5-(4-fluorophenyl)-1,2-oxazol-3-yl]met...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc(on2)-c2ccc(F)cc2)C1=O
Show InChI InChI=1S/C15H9FN2O4S2/c16-9-3-1-8(2-4-9)11-5-10(17-22-11)6-12-14(21)18(7-13(19)20)15(23)24-12/h1-6H,7H2,(H,19,20)/b12-6-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28904
PNG
(2-{5-[(3Z)-1-{[(3-methylphenyl)carbamoyl]methyl}-2...)
Show SMILES Cc1cccc(NC(=O)CN2C(=O)\C(=C3/SC(=S)N(CC(O)=O)C3=O)c3ccccc23)c1
Show InChI InChI=1S/C22H17N3O5S2/c1-12-5-4-6-13(9-12)23-16(26)10-24-15-8-3-2-7-14(15)18(20(24)29)19-21(30)25(11-17(27)28)22(31)32-19/h2-9H,10-11H2,1H3,(H,23,26)(H,27,28)/b19-18-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28904
PNG
(2-{5-[(3Z)-1-{[(3-methylphenyl)carbamoyl]methyl}-2...)
Show SMILES Cc1cccc(NC(=O)CN2C(=O)\C(=C3/SC(=S)N(CC(O)=O)C3=O)c3ccccc23)c1
Show InChI InChI=1S/C22H17N3O5S2/c1-12-5-4-6-13(9-12)23-16(26)10-24-15-8-3-2-7-14(15)18(20(24)29)19-21(30)25(11-17(27)28)22(31)32-19/h2-9H,10-11H2,1H3,(H,23,26)(H,27,28)/b19-18-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28896
PNG
(2-[(5Z)-5-{8-oxatricyclo[7.4.0.0^{2,7}]trideca-1(9...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cccc3c4ccccc4oc23)C1=O
Show InChI InChI=1S/C18H11NO4S2/c20-15(21)9-19-17(22)14(25-18(19)24)8-10-4-3-6-12-11-5-1-2-7-13(11)23-16(10)12/h1-8H,9H2,(H,20,21)/b14-8-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28895
PNG
(2-[(5Z)-5-[(2-methylquinolin-6-yl)methylidene]-4-o...)
Show SMILES Cc1ccc2cc(\C=C3/SC(=S)N(CC(O)=O)C3=O)ccc2n1
Show InChI InChI=1S/C16H12N2O3S2/c1-9-2-4-11-6-10(3-5-12(11)17-9)7-13-15(21)18(8-14(19)20)16(22)23-13/h2-7H,8H2,1H3,(H,19,20)/b13-7-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28894
PNG
(2-[(5Z)-5-(2H-1,3-benzodioxol-5-ylmethylidene)-4-o...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2ccc3OCOc3c2)C1=O
Show InChI InChI=1S/C13H9NO5S2/c15-11(16)5-14-12(17)10(21-13(14)20)4-7-1-2-8-9(3-7)19-6-18-8/h1-4H,5-6H2,(H,15,16)/b10-4-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28893
PNG
(2-[(5Z)-4-oxo-5-{[3-(1H-pyrazol-1-yl)phenyl]methyl...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cccc(c2)-n2cccn2)C1=O
Show InChI InChI=1S/C15H11N3O3S2/c19-13(20)9-17-14(21)12(23-15(17)22)8-10-3-1-4-11(7-10)18-6-2-5-16-18/h1-8H,9H2,(H,19,20)/b12-8-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28891
PNG
(2-[(5Z)-4-oxo-5-{[3-(pyrrolidin-1-yl)phenyl]methyl...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cccc(c2)N2CCCC2)C1=O
Show InChI InChI=1S/C16H16N2O3S2/c19-14(20)10-18-15(21)13(23-16(18)22)9-11-4-3-5-12(8-11)17-6-1-2-7-17/h3-5,8-9H,1-2,6-7,10H2,(H,19,20)/b13-9-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28890
PNG
(2-[(5Z)-4-oxo-5-[(4-phenylphenyl)methylidene]-2-su...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2ccc(cc2)-c2ccccc2)C1=O
Show InChI InChI=1S/C18H13NO3S2/c20-16(21)11-19-17(22)15(24-18(19)23)10-12-6-8-14(9-7-12)13-4-2-1-3-5-13/h1-10H,11H2,(H,20,21)/b15-10-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(Homo sapiens (Human))
BDBM28888
PNG
(2-[(5Z)-5-({7-bromo-2H,3H-thieno[3,4-b][1,4]dioxin...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2sc(Br)c3OCCOc23)C1=O
Show InChI InChI=1S/C12H8BrNO5S3/c13-10-9-8(18-1-2-19-9)5(21-10)3-6-11(17)14(4-7(15)16)12(20)22-6/h3H,1-2,4H2,(H,15,16)/b6-3-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28902
PNG
(2-[(5Z)-5-[(5-bromo-1H-indol-3-yl)methylidene]-4-o...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2c[nH]c3ccc(Br)cc23)C1=O
Show InChI InChI=1S/C14H9BrN2O3S2/c15-8-1-2-10-9(4-8)7(5-16-10)3-11-13(20)17(6-12(18)19)14(21)22-11/h1-5,16H,6H2,(H,18,19)/b11-3-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28901
PNG
(2-[(5Z)-5-(1H-indol-3-ylmethylidene)-4-oxo-2-sulfa...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2c[nH]c3ccccc23)C1=O
Show InChI InChI=1S/C14H10N2O3S2/c17-12(18)7-16-13(19)11(21-14(16)20)5-8-6-15-10-4-2-1-3-9(8)10/h1-6,15H,7H2,(H,17,18)/b11-5-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28900
PNG
(2-[(5Z)-4-oxo-2-sulfanylidene-5-{thieno[2,3-b]pyra...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cc3nccnc3s2)C1=O
Show InChI InChI=1S/C12H7N3O3S3/c16-9(17)5-15-11(18)8(21-12(15)19)4-6-3-7-10(20-6)14-2-1-13-7/h1-4H,5H2,(H,16,17)/b8-4-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28898
PNG
(2-[(5Z)-5-(1-benzothiophen-3-ylmethylidene)-4-oxo-...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2csc3ccccc23)C1=O
Show InChI InChI=1S/C14H9NO3S3/c16-12(17)6-15-13(18)11(21-14(15)19)5-8-7-20-10-4-2-1-3-9(8)10/h1-5,7H,6H2,(H,16,17)/b11-5-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28897
PNG
(2-[(5Z)-5-[(6-bromopyridin-2-yl)methylidene]-4-oxo...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cccc(Br)n2)C1=O
Show InChI InChI=1S/C11H7BrN2O3S2/c12-8-3-1-2-6(13-8)4-7-10(17)14(5-9(15)16)11(18)19-7/h1-4H,5H2,(H,15,16)/b7-4-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28896
PNG
(2-[(5Z)-5-{8-oxatricyclo[7.4.0.0^{2,7}]trideca-1(9...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2cccc3c4ccccc4oc23)C1=O
Show InChI InChI=1S/C18H11NO4S2/c20-15(21)9-19-17(22)14(25-18(19)24)8-10-4-3-6-12-11-5-1-2-7-13(11)23-16(10)12/h1-8H,9H2,(H,20,21)/b14-8-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
Collagenase


(homo sapiens (human))
BDBM28894
PNG
(2-[(5Z)-5-(2H-1,3-benzodioxol-5-ylmethylidene)-4-o...)
Show SMILES OC(=O)CN1C(=S)S\C(=C/c2ccc3OCOc3c2)C1=O
Show InChI InChI=1S/C13H9NO5S2/c15-11(16)5-14-12(17)10(21-13(14)20)4-7-1-2-8-9(3-7)19-6-18-8/h1-4H,5-6H2,(H,15,16)/b10-4-
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Burnham Institute for Medical Research



Assay Description
This assay was performed as outlined in the Anaspec MMP assay kit. The fluorescence peptide cleavage assay was performed in a 96-well plate in which ...


Chem Biol Drug Des 71: 131-9 (2008)


Article DOI: 10.1111/j.1747-0285.2007.00617.x
BindingDB Entry DOI: 10.7270/Q2KW5DCN
More data for this
Ligand-Target Pair
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